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Old 04-08-2010, 06:25 PM
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Default Superdrol/Methyldrostanolone

Superdrol/Methyldrostanolone

Androgenic Rating = 20

Anabolic Rating = 400

Chemical Name= 2a,17a-dimethyl-5a-androstane-17b-ol-3-one

Estrogenic Activity = none

Progestational Activity = no data available

Methyldrostanolone, also known as methasteron, is a potent oral anabolic steroid that was never sold as a prescription drug. In structure, this steroid is a close derivative of drostanolone (Masteron). The only difference in this case is the addition of a c-17 alpha methyl group, a modification that gives this steroid high oral bioavailability. The two agents remain very comparable, however. Both methyldrostanolone and drostanolone are non-aromatizable, so there is no difference in the estrogenicity of these two steroids, and both steroids retain favorable anabolic to androgenic ratios. Lab assays do put Superdrol ahead here, however, showing it to possess 4 times the anabolic potency of oral methyltestosterone while displaying only 20% of the androgenicity (a 20:1 ratio, compared to 3:1). The exact real-world relevance of these figures remains to be seen, however. Methyldrostanolone is favored by athletes for its moderate anabolic properties, which are usually accompanied by fat loss and minimal androgenic side effects.

History:
Methyldrostanolone was first described in 1959. This steroid was developed by the international pharmaceuticals giant Syntex, alongside such other well known anabolic agents as drostanolone propionate and Oxymetholone. Unlike drostanolone and oxymetholone, however, this steroid (at least in its basic form) was never released as a medicinal product. It was only sold for a brief period of time as a modified hormone called dimethazine. Dimethazine is made from two molecules of Methyldrostanolone that are bonded together, which are later metabolically separated to yield free Methyldrostanolone.

So while technically Methyldrostanolone itself was never sold as a prescription agent, we can say that the drug was one utilized medicinally.OtherWise, the methyldrostanolone molecule Methyldrostanolone remained an obscure research steroid only, and was never itself approved for use in humans. Methyldrostanolone was released in early 2005 as an over the counter "grey market" anabolic steroid in the United States.

The drug was being sold without restrictions as a nutritional supplement product, barring some minimum age disclaimers by the manufacturer. No State or Federal laws identify this drug as an anabolic steroid, which remove the legalities associated with being a Class III controlled substance like other steroids. This is simply due to the fact that methyldrostanolone was not in commerce at the time such laws were written, and was unknown to lawmakers. It was never legal to sell as a dietary supplement, however, and in late 2005 the FDA angrily acknowledged methyldrostanolone was being sold on the sports supplement market. In early 2006, the FDA sent letters to the manufacturer and a distributor demanding it be pulled from commerce. Superdrol has since been discontinued.

Structural Characteristics:
Methyldrostanolone is a modified form of dihydrotestosterone. It differs by: 1) the addition of a methyl group at carbon 17-alpha, which helps protect the hormone during oral administration, and 2) the introduction of a methyl group at carbon-2 (alpha), which considerably increases the anabolic strength of the steroid by heightening its resistance to metabolism by the 3-hydroxysteroid dehydrogenase enzyme in skeletal muscle tissue.

Side Effects (Estrogenic):
Methyldrostanolone is not aromatized by the body, and is not measurably estrogenic. An anti-estrogen is not necessary when using this steroid, as gynecomastia should not be a concern even among sensitive individuals. Since estrogen is the usual culprit with water retention, methyldrostanolone instead produces a lean, quality look to the physique with no fear of excess subcutaneous fluid retention. This makes it a favorable steroid to use during cutting cycles, when water and fat retention are major concerns.

Administration (Men):
Methydrostanolone was never approved for use in humans. Prescribing guidelines are unavailable. An effective dosage of methyldrostanolone for physique or performance-enhancing purposes seems to begin in the range of 10-20 mg per day, taken for no longer than 6 or 8 weeks. At this level it seems to impart a measurable muscle-building effect, which is usually accompanied by fat loss and increased definition. Don't expect to gain 30 pounds on this agent (its name, which is short for "Super Anadrol" is more marketing than reality), but many do walk away with more than 10 pounds of solid muscle gain when using this agent alone. In determining an optimal daily dosage, some do find the drug to be measurably more effective when venturing up to the 30 mg range. Potential hepatotoxicity should definitely be taken into account with such use, however.

To avoid further escalating liver strain, 20 mg daily of daily of methyldrostanolone is sometimes stacked with a non-toxic injectable steroid, such as testosterone for mass-building phases of training, or nandrolone or boldenone for more lean tissue gain and definition, instead of simply increasing the dosage.The drug also works well in cutting cycles,where its lack of estrogenicity is highly favored. Often it is combined here with a non-aromatizable Injectable steroid like Primobolan or Parabolan.

Administration (Women):
Methyldrostanolone was never approved for use in humans. Prescribing guidelines are unavailable. In the athletic arena, an effective oral daily dosage would fall around 2.5 mg per day, taken in cycles lasting no more fhan 4-6 weeks to minimize the chance for virilization. The main point of contention with females is probably going to be the 10 mg per capsule dosage, which is far too high to use. Application would require opening each capsule and splitting the powdered contents up into 4 separate doses. As with all steroids, virilization is still possible.

Availability:
Superdrol is no longer commercially produced, although some clone products may still be located.

This is not my original work, credit goes to William Llewellyn and his book Anabolics 2009.
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Old 04-16-2010, 05:50 PM
Bonaparte Bonaparte is offline
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Superdrol is much more androgenic in vivo than its numbers suggest.
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Old 04-24-2010, 04:00 PM
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Superdrol is much more androgenic in vivo than its numbers suggest.
It is one of the few steroids that has no affinity for SHBG, so I agree with you on that.
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Old 04-24-2010, 04:06 PM
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great read! i have been waiting for this lol! good find
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Old 04-25-2010, 01:04 PM
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i heard somewhere that superdrol leads to loss of libido. just wanted to confirm if it does.
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Old 04-25-2010, 01:28 PM
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i heard somewhere that superdrol leads to loss of libido. just wanted to confirm if it does.
it did about 3 weeks into the cycle. before that i was fine, but then it hit me. this was when i ran sd by itself, not with test. never run it without test imho!
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Old 04-25-2010, 03:25 PM
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great read! i have been waiting for this lol! good find
No problem bro, always happy to provide good information whenever I can!
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Old 04-25-2010, 05:08 PM
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we should get a good m1t in here also
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Old 03-26-2011, 10:26 AM
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Originally Posted by Grow-bot View Post
It is one of the few steroids that has no affinity for SHBG, so I agree with you on that.
I keep trying to find some proof of this, but haven't been successful. In fact most write-ups on it say the exact opposite that shbg binds strongly to SD. Does someone have a link or maybe have a little explanation if the statement above is true? I'd like to believe that it's true
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Old 03-26-2011, 12:47 PM
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Glad i stocked up on Methadrol and M1T both 10 and 5 mg pills, both give great results and lean gains for me
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Old 03-29-2011, 03:06 PM
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I keep trying to find some proof of this, but haven't been successful. In fact most write-ups on it say the exact opposite that shbg binds strongly to SD. Does someone have a link or maybe have a little explanation if the statement above is true? I'd like to believe that it's true
I read this somewhere, but cannot find it now. All the other write-ups point to a high affinity for SHBG, which seems strange to me. If it does have a high affinity for SHBG, why does one require such a small amount of it to make explosive gains? I can believe highly suppressive, but not highly binding.

Any AAS that I have used that have a strong affinity for SHBG (supposedly anyway) required dosages in the hundreds of mgs daily range to work effectively.

MENT for example has almost no affinity for SHBG and most people can get great gains off of 50mgs EOD.

I'll keep looking and admittedly it would not be the first time that some data I picked up was wrong.

Another conclusion is that if Superdrol has a high affinity for SBHG, and it still imparts the gains that it can, then unbound Superdrol is a VERY powerful AAS. Note that Proviron, DHT, and Mestanolone have a high binding affinity for SBHG and I have yet to hear of one person saying that they got massive off of a cycle of any of these.
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Old 03-29-2011, 08:23 PM
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I loved C's superdrol!!!!!
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Old 03-30-2011, 09:37 PM
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Quote:
Originally Posted by Grow-bot View Post
I read this somewhere, but cannot find it now. All the other write-ups point to a high affinity for SHBG, which seems strange to me. If it does have a high affinity for SHBG, why does one require such a small amount of it to make explosive gains? I can believe highly suppressive, but not highly binding.

Any AAS that I have used that have a strong affinity for SHBG (supposedly anyway) required dosages in the hundreds of mgs daily range to work effectively.

MENT for example has almost no affinity for SHBG and most people can get great gains off of 50mgs EOD.

I'll keep looking and admittedly it would not be the first time that some data I picked up was wrong.

Another conclusion is that if Superdrol has a high affinity for SBHG, and it still imparts the gains that it can, then unbound Superdrol is a VERY powerful AAS. Note that Proviron, DHT, and Mestanolone have a high binding affinity for SBHG and I have yet to hear of one person saying that they got massive off of a cycle of any of these.
Good point. I could agree with your reasoning.
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Old 08-25-2012, 03:04 AM
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Do you even lift
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Old 01-12-2015, 03:31 PM
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love this place still after all these years
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Old 06-03-2015, 08:32 PM
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Ill pass on stuff like superdrol

It was rejected by pharmacy for a reason

Much better and safer options are available

Imho.... stick with orals that were pharmacy approved

Not ones that were on the reject list

Think about it ......
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Old 06-06-2015, 10:08 PM
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superdrol was insane. I looked amazing on it however, but was a nervous tweaker with high BP. Even at very low doses like 2.5mg day I could still feel the effects. Gave the muscles a very dry grainy look but still full.
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Old 06-11-2015, 12:30 AM
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Quote:
Originally Posted by Mack View Post
Ill pass on stuff like superdrol

It was rejected by pharmacy for a reason

Much better and safer options are available

Imho.... stick with orals that were pharmacy approved

Not ones that were on the reject list

Think about it ......
Your not wrong in your logic. ADROL has fewer sides and generally more results. Imagine that, Adrol safer than ANYTHING? Its easier on your liver for sure. (not that its easy at all though).
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Old 06-19-2018, 01:25 PM
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Quote:
Originally Posted by Mack View Post
Ill pass on stuff like superdrol

It was rejected by pharmacy for a reason

Much better and safer options are available

Imho.... stick with orals that were pharmacy approved

Not ones that were on the reject list

Think about it ......

Exactly. I've taken just about ever steroid there is and superdrol made me feel lethargic as all hell.
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Old 07-04-2018, 07:18 PM
Xxplosive Xxplosive is offline
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Quote:
Originally Posted by Mack View Post
Ill pass on stuff like superdrol

It was rejected by pharmacy for a reason

Much better and safer options are available

Imho.... stick with orals that were pharmacy approved

Not ones that were on the reject list

Think about it ......
Nothing cuts, adds size, increases vascularity like superdrol.

Pharms likely passed on it bc it doesnt provide any real medical purposes.

The only thing that compares is primo... which is a lot more expensive.

IMHO, superdrol is less toxic than tren, which most swear by. I was shitting blood at one point on tren. Worst thing superdrol ever did was make me a bit lethargic, and even then i think thats just if you over do it. I actually would get a rush of energy/euphoria for the first hour or two when i used injectable superdrol.

I will be giving my first run of oral sdrol here starting in about a week.
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Old 10-03-2018, 04:31 AM
tmikes tmikes is online now
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Quote:
Originally Posted by Xxplosive View Post
Nothing cuts, adds size, increases vascularity like superdrol.

Pharms likely passed on it bc it doesnt provide any real medical purposes.

The only thing that compares is primo... which is a lot more expensive.

IMHO, superdrol is less toxic than tren, which most swear by. I was shitting blood at one point on tren. Worst thing superdrol ever did was make me a bit lethargic, and even then i think thats just if you over do it. I actually would get a rush of energy/euphoria for the first hour or two when i used injectable superdrol.

I will be giving my first run of oral sdrol here starting in about a week.
Xx,

Checking in to see how the superdrol was going. What’s been your results so far? How long can you take it for? I have some on hand and will be using it in the future. First time.

Thanks.
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Old 10-09-2018, 09:56 PM
Xxplosive Xxplosive is offline
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Xx,

Checking in to see how the superdrol was going. What’s been your results so far? How long can you take it for? I have some on hand and will be using it in the future. First time.

Thanks.
If you are gonna run it... Find an injectable version. I did oral for the first time, and while it was super effective, it really does tax the fuck out of you and makes you feel like shit after a few weeks.

That 1 less pass through the liver and not needing to use as much goes a long way in not just your health, but effectiveness- what good is a compound that makes you feel so shitty its a drag to train?
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  #23  
Old 06-18-2018, 09:40 PM
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Can't wait to start my Sdrol cycle

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